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▷ Pioglitazona: ¿Qué es y para qué sirve? - Todo sobre medicamentos Ir al Contenido La Pioglitazona es útil para el tratamiento de la diabetes tipo 2 , es decir, aquella donde el cuerpo no puede usar de forma normal la insulina que produce y por lo cual, no se regulan los niveles de glucosa en sangre.
Este medicamento funciona de mejor manera al ser acompañado por un régimen de buena alimentación y ejercicio.
¿Cómo funciona la Pioglitazona ? Este medicamento funciona aumentando la sensibilidad del cuerpo a la insulina de células hepáticas, tejido adiposo y músculo esquelético. La glucosa se absorbe de mejor manera y produce energía.
La absorción de Pioglitazona se realiza de forma rápida, teniendo su pico máximo a las 2 horas de ser ingerido. Si es consumido con comidas este pico puede tardar una hora más.
Este medicamento puede combinarse con Metformina, Sulfonilurea o Insulina y esto depende de la tolerancia de cada paciente a las sustancias activas.
Recuerde que la diabetes bien tratada evita la posibilidad de que sufra infartos, apoplejía, deficiencia renal, daño en los nervios o problemas de la vista
Dosis de Pioglitazona La vía de administración de este medicamento es oral.
La dosis recomendada es de 1 vez al día con o sin comidas .
Se puede iniciar con 15 o 30mg y aumentar hasta 45mg por día.
Cabe señalar que Pioglitazona sólo controla la enfermedad, no la cura.
Pioglitazona con dieta y ejercicio Como en toda persona que padece de diabetes, la sugerencia de llevar una dieta saludable es esencial. El sobrepeso o la obesidad sólo harán que su bienestar se vea comprometido y pueda terminar en la muerte.
Asimismo, el hábito del ejercicio físico abonará a que el medicamento funcione de mejor manera.
Pioglitazona y Alcohol La ingesta de alcohol no está recomendada en pacientes con diabetes , ya que éste puede ocasionar la disminución de azúcar en la sangre (hipoglucemia). Usted puede consultar con su médico las instrucciones que debe seguir para el consumo de este tipo de bebidas.
Pioglitazona y Metformina Es posible que su médico considere la opción de usar una combinación de Pioglitazona y Metformina para tratar su diabetes.
Por un lado, la Pioglitazona ayudará a su organismo a ser más sensible a la insulina, por lo que la regulación de glucosa se hace de mejor manera.
Por otro lado, la Metformina actúa disminuyendo la producción de glucosa por parte del hígado.
Si quieres conocer qué otros usos tiene la Metformina, revisa Metformina para adelgazar .
Contraindicaciones y Riesgos de Pioglitazona Al iniciar con un tratamiento de diabetes, se debe considerar el listado de padecimientos o factores de riesgo que se tienen para acceder a la medicina que se nos recete. Para la Pioglitazona, el listado de advertencias es amplio y debe ser estudiado por médico y paciente. Revise las siguientes precauciones.
La Pioglitazona puede causar o empeorar una insuficiencia cardiaca, debe avisar a su médico sobre su historial. Informar al médico si ha tenido inflamación de brazos, manos pies, tobillos o piernas Notificar si tiene niveles altos de colesterol o grasas en la sangre o presión arterial alta Si tiene apnea del sueño, hablar con su médico Pioglitazona no está indicada para embarazo o lactancia Pioglitazona puede aumentar las posibilidades de quedar embarazada, por lo cual su médico le recomendará exámenes frecuentes. Si tiene hipersensibilidad a la sustancia no está indicado Evitar este medicamento en personas con insuficiencia hepática Evitar este medicamento en personas con cáncer de vejiga Efectos secundarios de Pioglitazona Para iniciar, usted debe ser consciente de que este medicamento puede causar cambios en su nivel de azúcar, por lo cual, el monitoreo constante es indispensable para que no sufra ningún incidente de salud. Aunado a ello, los efectos adversos que puede tener son variados y debe acudir a su médico en caso de que se agraven o sean constantes.
Aumento de peso Infecciones respiratorias Alteraciones de la visión Gases Cefaleas En combinación con Metformina
Anemia Dolor de cabeza Disfunción eréctil Alteraciones de la visión Artralgia En combinación con otros medicamentos como sulfonilurea o insulina, pueden añadirse variedad de efectos adversos.
De igual manera, este producto puede producir problemas hepáticos. También, en estudios se comprobó el desarrollo de cáncer de vejiga en hombres y mujeres y aumento de fracturas de manos, brazos o pies en mujeres
¿Cuánto cuesta y dónde puedo comprar Pioglitazona? En el mercado puedes encontrar este medicamento por su nombre genérico o por nombres comerciales como Glitacar 1 o Zactos. Revisa sus precios.
Pioglitazona (Genérico) Caja con 7 tabletas de 30mg. Su precio oscila entre 25 y 40 pesos mexicanos. Glitacar 1 Caja con 7 tabletas de 15mg. Su precio oscila entre 200 y 300 pesos mexicanos. Caja con 30 tabletas de 15mg. Su precio oscila entre 700 y 750 pesos mexicanos. Caja con 30 tabletas de 30mg. Su precio oscila entre 1200 y 1300 pesos mexicanos. Zactos Caja con 7 tabletas de 40mg. Su precio oscila entre 700 y 900 pesos mexicanos Caja con 28 tabletas de 15mg. Su precio oscila entre 1200 y 1300 pesos mexicanos Caja con 28 tabletas de 30mg. Su precio oscila entre 2200 y 2300 pesos mexicanos Recuerda que puedes adquirir Pioglitazona (Genérico), Glitacar 1 y Zactos en Farmacias Prixz, Farmacias Benavides, Farmacias San Pablo, entre otras.
¿Qué es la Pioglitazona? La pioglizona es un medicamento que sirve como tratamiento de la diabetes mellitus tipo 2 se puede administrar por vía oral solo o en combinación con otros fármacos
Pertenece a la familia de las tiazolidinedionas por lo que está emparentado con otros medicamentos de este grupo terapéutico como la rosiglotazona y la troglitazona.
¿Cuál es su mecanismo de acción de Pioglitazona? La Pioglitazona aumenta la sensibilidad de la insulina, en las células musculares y las células que forman el tejido adiposo. Al ser la insulina contribuyen al descenso de glucosa en sangre, el efecto final de la pioglitazona es también hipoglucemiante. La acción del fármaco se basa en su unión a un receptor celular conocido como receptor gamma activado por el proliferador de peroxisomas, esta unión provoca la activación de varios genes que promueven o facilitan las acciones de la insulina. Además de este efecto, causa una reducción en la producción de glucosa por las células del hígado.
Solo es eficaz en aquellos pacientes que muestran un nivel adecuado de insulina en sangre.
¿Presentaciones y dosis de Pioglitazona? Se administra por vía oral en forma de comprimidos, a una dosis comprendida entre 15 y 45 mg al día, se puede acompañar con o sin alimento. Se deben tragar los comprimidos con un vaso de agua.
Se venden regularmente en pastillas de 15 mg o 30 mg bajo patentes como Gliozac, Zactos, entre otras.
¿Cuáles son las advertencias y contraindicaciones de Pioglitazona? Antes de iniciar tratamiento con pioglitazona se deben valorar los siguientes factores:
Riesgo de cáncer de vejiga (los causantes pueden ser; la edad, antecedente de tabaquismo, exposición a agentes quimioterápicos como ciclofosfamida o radioterapia previa en zona pélvica) Se debera descartar hematuria macroscópica Se deberá valorar respuesta con el medicamente de 3 a 6 meses y si no se ven cambios beneficiosos suspender el tratamiento y continuar revisiones rutinarias para confirmar beneficio ante los riesgos del tratamiento prolongado. Personas con factor de riesgo infarto de miocardio se deberá notificar al medico Empezar con dosis mín. posible y aumentar gradualmente. Vigilar signos de insuficiencia cardiaca, aumento de peso y edema, especialmente con disminución de reserva cardiaca, asociado con insulina y con historial de insuficiencia cardiaca se deberá suspender el tratamiento si hay empeoramiento de función cardiaca. En personas de edad avanzada se deberá tener mayor precaución Es importante avisar al médico si esta en procesos de embarazo o lactancia para que le de las indicaciones adecuadas ya que no hay muchos estudios que corroboren si es apto para mujeres en esta situación ¿Cuáles son los efectos secundarios de Pioglitazona? Puede provocar algunos efectos secundarios como los siguientes :
Insuficiencia cardíaca por retención de líquidos Aumenta la probabilidad de aparición de cáncer de vejiga, motivo por el que se ha prohibido en algunos países. Provocación de edema que aunque generalmente es leve Puede causar la descompensación de una insuficiencia cardíaca que existía antes del inicio del tratamiento. En el 2% de los pacientes tratados provoca lesión hepática que generalmente es de carácter leve Infecciones tracto respiratorio superior aumento de peso hipoestesia fractura ósea Anomalías de visión ¿Dónde comprar y qué precio tiene Pioglitazona? Lo puedes comprar en establecimientos en México como: Farmacias del ahorro, Farmacias San Pablo, chedrahui, Walmart, Farmacias similares, entre otros.
La pioglitazona la podrás comprar a un precio generalmente que oscila entre los $130 hasta los $200 pesos dependiendo si es de patente o genérico.